Fluorine in PDB 7jn3: Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048

Enzymatic activity of Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048

All present enzymatic activity of Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048:
2.7.7.49; 2.7.7.7; 3.1.26.4;

Other elements in 7jn3:

The structure of Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048 also contains other interesting chemical elements:

Zinc (Zn) 2 atoms
Magnesium (Mg) 4 atoms
Chlorine (Cl) 2 atoms

Fluorine Binding Sites:

The binding sites of Fluorine atom in the Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048 (pdb code 7jn3). This binding sites where shown within 5.0 Angstroms radius around Fluorine atom.
In total 2 binding sites of Fluorine where determined in the Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048, PDB code: 7jn3:
Jump to Fluorine binding site number: 1; 2;

Fluorine binding site 1 out of 2 in 7jn3

Go back to Fluorine Binding Sites List in 7jn3
Fluorine binding site 1 out of 2 in the Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048


Mono view


Stereo pair view

A full contact list of Fluorine with other atoms in the F binding site number 1 of Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048 within 5.0Å range:
probe atom residue distance (Å) B Occ
A:F302

b:53.6
occ:1.00
FAH A:ZZX302 0.0 53.6 1.0
CAT A:ZZX302 1.3 53.6 1.0
CAV A:ZZX302 2.4 53.6 1.0
CAJ A:ZZX302 2.4 53.6 1.0
CLAI A:ZZX302 2.9 53.6 1.0
CG A:GLN151 3.2 52.2 1.0
CAK A:ZZX302 3.6 53.6 1.0
CAL A:ZZX302 3.6 53.6 1.0
N2 I:DG4 3.8 44.5 1.0
C2 I:DG4 3.9 44.5 1.0
N1 I:DG4 3.9 44.5 1.0
CB A:GLN151 4.0 52.2 1.0
CAU A:ZZX302 4.1 53.6 1.0
O A:SER150 4.3 51.5 1.0
CD A:GLN151 4.3 52.2 1.0
NE2 A:GLN151 4.4 52.2 1.0
CA A:GLN151 4.4 52.2 1.0
N4 J:DC35 4.5 52.3 1.0
N3 I:DG4 4.5 44.5 1.0
C6 I:DG4 4.5 44.5 1.0
C4 J:DC35 4.6 52.3 1.0
C5 J:DC35 4.7 52.3 1.0
C A:SER150 4.9 51.5 1.0

Fluorine binding site 2 out of 2 in 7jn3

Go back to Fluorine Binding Sites List in 7jn3
Fluorine binding site 2 out of 2 in the Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048


Mono view


Stereo pair view

A full contact list of Fluorine with other atoms in the F binding site number 2 of Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048 within 5.0Å range:
probe atom residue distance (Å) B Occ
E:F302

b:69.2
occ:1.00
FAH E:ZZX302 0.0 69.2 1.0
CAT E:ZZX302 1.4 69.2 1.0
CAV E:ZZX302 2.4 69.2 1.0
CAJ E:ZZX302 2.4 69.2 1.0
CLAI E:ZZX302 2.9 69.2 1.0
CG E:GLN151 3.3 55.5 1.0
N2 K:DG4 3.5 98.0 1.0
N1 K:DG4 3.6 98.0 1.0
C2 K:DG4 3.6 98.0 1.0
CAL E:ZZX302 3.6 69.2 1.0
CAK E:ZZX302 3.6 69.2 1.0
CB E:GLN151 4.0 55.5 1.0
N4 L:DC35 4.0 59.4 1.0
CAU E:ZZX302 4.1 69.2 1.0
O E:SER150 4.2 60.8 1.0
C4 L:DC35 4.3 59.4 1.0
CA E:GLN151 4.3 55.5 1.0
C6 K:DG4 4.3 98.0 1.0
N3 K:DG4 4.4 98.0 1.0
C5 L:DC35 4.5 59.4 1.0
CD E:GLN151 4.6 55.5 1.0
NE2 E:GLN151 4.7 55.5 1.0
O6 K:DG4 4.8 98.0 1.0
N3 L:DC35 4.8 59.4 1.0
C E:SER150 4.8 60.8 1.0
C4 K:DG4 5.0 98.0 1.0

Reference:

K.K.Pandey, S.Bera, K.Shi, H.Aihara, D.P.Grandgenett, M.J.Rau, A.V.Oleru, J.A.J.Fitzpatrick, A.N.Engelman. Cryo-Em Structure of Rous Sarcoma Virus Cleaved Synaptic Complex (Csc) with Hiv-1 Integrase Strand Transfer Inhibitor Mk-2048 Commun Biol 2021.
ISSN: ESSN 2399-3642
DOI: 10.1038/S42003-021-01855-2
Page generated: Sat Apr 3 15:09:25 2021

Last articles

Zn in 8WB0
Zn in 8WAX
Zn in 8WAU
Zn in 8WAZ
Zn in 8WAY
Zn in 8WAV
Zn in 8WAW
Zn in 8WAT
Zn in 8W7M
Zn in 8WD3
© Copyright 2008-2020 by atomistry.com
Home   |    Site Map   |    Copyright   |    Contact us   |    Privacy