|
Fluorine in PDB 7yi7: Crystal Structure of Human HPSE1 in Complex with InhibitorEnzymatic activity of Crystal Structure of Human HPSE1 in Complex with Inhibitor
All present enzymatic activity of Crystal Structure of Human HPSE1 in Complex with Inhibitor:
3.2.1.166; Protein crystallography data
The structure of Crystal Structure of Human HPSE1 in Complex with Inhibitor, PDB code: 7yi7
was solved by
M.Mima,
N.Fujimoto,
Y.Imai,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Fluorine Binding Sites:
The binding sites of Fluorine atom in the Crystal Structure of Human HPSE1 in Complex with Inhibitor
(pdb code 7yi7). This binding sites where shown within
5.0 Angstroms radius around Fluorine atom.
In total 3 binding sites of Fluorine where determined in the Crystal Structure of Human HPSE1 in Complex with Inhibitor, PDB code: 7yi7: Jump to Fluorine binding site number: 1; 2; 3; Fluorine binding site 1 out of 3 in 7yi7Go back to Fluorine Binding Sites List in 7yi7
Fluorine binding site 1 out
of 3 in the Crystal Structure of Human HPSE1 in Complex with Inhibitor
Mono view Stereo pair view
Fluorine binding site 2 out of 3 in 7yi7Go back to Fluorine Binding Sites List in 7yi7
Fluorine binding site 2 out
of 3 in the Crystal Structure of Human HPSE1 in Complex with Inhibitor
Mono view Stereo pair view
Fluorine binding site 3 out of 3 in 7yi7Go back to Fluorine Binding Sites List in 7yi7
Fluorine binding site 3 out
of 3 in the Crystal Structure of Human HPSE1 in Complex with Inhibitor
Mono view Stereo pair view
Reference:
Y.Imai,
D.Wakasugi,
R.Suzuki,
S.Kato,
M.Sugisaki,
M.Mima,
H.Miyagawa,
M.Endo,
N.Fujimoto,
T.Fukunaga,
S.Kato,
S.Kuroda,
T.Takahashi,
H.Kakinuma.
Lead Identification of Novel Tetrahydroimidazo[1,2-A]Pyridine-5-Carboxylic Acid Derivative As A Potent Heparanase-1 Inhibitor. Bioorg.Med.Chem.Lett. V. 79 29050 2022.
Page generated: Wed Apr 5 01:53:40 2023
ISSN: ESSN 1464-3405 PubMed: 36368497 DOI: 10.1016/J.BMCL.2022.129050 |
Last articlesZn in 8WB0Zn in 8WAX Zn in 8WAU Zn in 8WAZ Zn in 8WAY Zn in 8WAV Zn in 8WAW Zn in 8WAT Zn in 8W7M Zn in 8WD3 |
© Copyright 2008-2020 by atomistry.com | ||
Home | Site Map | Copyright | Contact us | Privacy |