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Atomistry » Fluorine » PDB 8pgi-8py3 » 8pqh » |
Fluorine in PDB 8pqh: Pdgfra T674I Mutant Kinase Domain in Complex with AvapritinibEnzymatic activity of Pdgfra T674I Mutant Kinase Domain in Complex with Avapritinib
All present enzymatic activity of Pdgfra T674I Mutant Kinase Domain in Complex with Avapritinib:
2.7.10.1; Protein crystallography data
The structure of Pdgfra T674I Mutant Kinase Domain in Complex with Avapritinib, PDB code: 8pqh
was solved by
A.Teuber,
S.Kleinboelting,
M.P.Mueller,
D.Rauh,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Fluorine Binding Sites:
The binding sites of Fluorine atom in the Pdgfra T674I Mutant Kinase Domain in Complex with Avapritinib
(pdb code 8pqh). This binding sites where shown within
5.0 Angstroms radius around Fluorine atom.
In total only one binding site of Fluorine was determined in the Pdgfra T674I Mutant Kinase Domain in Complex with Avapritinib, PDB code: 8pqh: Fluorine binding site 1 out of 1 in 8pqhGo back to Fluorine Binding Sites List in 8pqh
Fluorine binding site 1 out
of 1 in the Pdgfra T674I Mutant Kinase Domain in Complex with Avapritinib
Mono view Stereo pair view
Reference:
A.Teuber,
T.Schulz,
B.S.Fletcher,
R.Gontla,
T.Muehlenberg,
M.-L.Zischinsky,
J.Niggenaber,
J.Weisner,
S.B.Kleinboelting,
J.Lategahn,
S.Sievers,
M.P.Mueller,
S.Bauer,
D.Rauh.
Avapritinib-Based Sar Studies Reveal A Binding Pocket in Kit and Pdgfra Nat Commun 2023.
Page generated: Fri Aug 2 22:20:51 2024
ISSN: ESSN 2041-1723 DOI: 10.1038/S41467-023-44376-8 |
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