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Atomistry » Fluorine » PDB 3uyt-3vrb » 3vf8 » |
Fluorine in PDB 3vf8: Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416Enzymatic activity of Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416
All present enzymatic activity of Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416:
2.7.10.2; Protein crystallography data
The structure of Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416, PDB code: 3vf8
was solved by
L.R.Mclean,
Y.Zhang,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Fluorine Binding Sites:
The binding sites of Fluorine atom in the Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416
(pdb code 3vf8). This binding sites where shown within
5.0 Angstroms radius around Fluorine atom.
In total only one binding site of Fluorine was determined in the Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416, PDB code: 3vf8: Fluorine binding site 1 out of 1 in 3vf8Go back to![]() ![]()
Fluorine binding site 1 out
of 1 in the Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416
![]() Mono view ![]() Stereo pair view
Reference:
L.R.Mclean,
Y.Zhang,
N.Zaidi,
X.Bi,
R.Wang,
R.Dharanipragada,
J.G.Jurcak,
T.A.Gillespy,
Z.Zhao,
K.Y.Musick,
Y.M.Choi,
M.Barrague,
J.Peppard,
M.Smicker,
M.Duguid,
A.Parkar,
J.Fordham,
D.Kominos.
X-Ray Crystallographic Structure-Based Design of Selective Thienopyrazole Inhibitors For Interleukin-2-Inducible Tyrosine Kinase. Bioorg.Med.Chem.Lett. V. 22 3296 2012.
Page generated: Mon Jul 14 19:53:04 2025
ISSN: ISSN 0960-894X PubMed: 22464456 DOI: 10.1016/J.BMCL.2012.03.016 |
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