|
Atomistry » Fluorine » PDB 3uyt-3vrb » 3vf8 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Atomistry » Fluorine » PDB 3uyt-3vrb » 3vf8 » |
Fluorine in PDB 3vf8: Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416Enzymatic activity of Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416
All present enzymatic activity of Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416:
2.7.10.2; Protein crystallography data
The structure of Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416, PDB code: 3vf8
was solved by
L.R.Mclean,
Y.Zhang,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Fluorine Binding Sites:
The binding sites of Fluorine atom in the Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416
(pdb code 3vf8). This binding sites where shown within
5.0 Angstroms radius around Fluorine atom.
In total only one binding site of Fluorine was determined in the Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416, PDB code: 3vf8: Fluorine binding site 1 out of 1 in 3vf8Go back to Fluorine Binding Sites List in 3vf8
Fluorine binding site 1 out
of 1 in the Crystal Structure of Spleen Tyrosine Kinase Syk Catalytic Domain with Pyrazolylbenzimidazole Inhibitor 416
Mono view Stereo pair view
Reference:
L.R.Mclean,
Y.Zhang,
N.Zaidi,
X.Bi,
R.Wang,
R.Dharanipragada,
J.G.Jurcak,
T.A.Gillespy,
Z.Zhao,
K.Y.Musick,
Y.M.Choi,
M.Barrague,
J.Peppard,
M.Smicker,
M.Duguid,
A.Parkar,
J.Fordham,
D.Kominos.
X-Ray Crystallographic Structure-Based Design of Selective Thienopyrazole Inhibitors For Interleukin-2-Inducible Tyrosine Kinase. Bioorg.Med.Chem.Lett. V. 22 3296 2012.
Page generated: Sun Dec 13 11:57:01 2020
ISSN: ISSN 0960-894X PubMed: 22464456 DOI: 10.1016/J.BMCL.2012.03.016 |
Last articlesZn in 8WB0Zn in 8WAX Zn in 8WAU Zn in 8WAZ Zn in 8WAY Zn in 8WAV Zn in 8WAW Zn in 8WAT Zn in 8W7M Zn in 8WD3 |
© Copyright 2008-2020 by atomistry.com | ||
Home | Site Map | Copyright | Contact us | Privacy |