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Atomistry » Fluorine » PDB 5wfo-5xd5 » 5wg4 » |
Fluorine in PDB 5wg4: Human GRK2 in Complex with Gbetagamma Subunits and CCG257284Enzymatic activity of Human GRK2 in Complex with Gbetagamma Subunits and CCG257284
All present enzymatic activity of Human GRK2 in Complex with Gbetagamma Subunits and CCG257284:
2.7.11.15; Protein crystallography data
The structure of Human GRK2 in Complex with Gbetagamma Subunits and CCG257284, PDB code: 5wg4
was solved by
R.Bouley,
J.J.G.Tesmer,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Fluorine Binding Sites:
The binding sites of Fluorine atom in the Human GRK2 in Complex with Gbetagamma Subunits and CCG257284
(pdb code 5wg4). This binding sites where shown within
5.0 Angstroms radius around Fluorine atom.
In total only one binding site of Fluorine was determined in the Human GRK2 in Complex with Gbetagamma Subunits and CCG257284, PDB code: 5wg4: Fluorine binding site 1 out of 1 in 5wg4Go back to![]() ![]()
Fluorine binding site 1 out
of 1 in the Human GRK2 in Complex with Gbetagamma Subunits and CCG257284
![]() Mono view ![]() Stereo pair view
Reference:
R.Bouley,
H.V.Waldschmidt,
M.C.Cato,
A.Cannavo,
J.Song,
J.Y.Cheung,
X.Q.Yao,
W.J.Koch,
S.D.Larsen,
J.J.G.Tesmer.
Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors. Mol. Pharmacol. V. 92 707 2017.
Page generated: Tue Jul 15 08:59:46 2025
ISSN: ESSN 1521-0111 PubMed: 29070696 DOI: 10.1124/MOL.117.110130 |
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