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Atomistry » Fluorine » PDB 7tsd-7u8s » 7ty2 | ||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Atomistry » Fluorine » PDB 7tsd-7u8s » 7ty2 » |
Fluorine in PDB 7ty2: Crystal Structure of SETD2 Bound to An Indole-Based InhibitorEnzymatic activity of Crystal Structure of SETD2 Bound to An Indole-Based Inhibitor
All present enzymatic activity of Crystal Structure of SETD2 Bound to An Indole-Based Inhibitor:
2.1.1.359; Protein crystallography data
The structure of Crystal Structure of SETD2 Bound to An Indole-Based Inhibitor, PDB code: 7ty2
was solved by
N.A.Farrow,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Other elements in 7ty2:
The structure of Crystal Structure of SETD2 Bound to An Indole-Based Inhibitor also contains other interesting chemical elements:
Fluorine Binding Sites:
The binding sites of Fluorine atom in the Crystal Structure of SETD2 Bound to An Indole-Based Inhibitor
(pdb code 7ty2). This binding sites where shown within
5.0 Angstroms radius around Fluorine atom.
In total only one binding site of Fluorine was determined in the Crystal Structure of SETD2 Bound to An Indole-Based Inhibitor, PDB code: 7ty2: Fluorine binding site 1 out of 1 in 7ty2Go back to![]() ![]()
Fluorine binding site 1 out
of 1 in the Crystal Structure of SETD2 Bound to An Indole-Based Inhibitor
![]() Mono view ![]() Stereo pair view
Reference:
J.S.Alford,
J.W.Lampe,
D.Brach,
R.Chesworth,
K.Cosmopoulos,
K.W.Duncan,
S.T.Eckley,
J.L.Kutok,
A.Raimondi,
T.V.Riera,
B.Shook,
C.Tang,
J.Totman,
N.A.Farrow.
Conformational-Design-Driven Discovery of EZM0414: A Selective, Potent SETD2 Inhibitor For Clinical Studies. Acs Med.Chem.Lett. V. 13 1137 2022.
Page generated: Wed Jul 16 00:42:47 2025
ISSN: ISSN 1948-5875 PubMed: 35859865 DOI: 10.1021/ACSMEDCHEMLETT.2C00167 |
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