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Atomistry » Fluorine » PDB 5btf-5cgq » 5bvn » |
Fluorine in PDB 5bvn: Fragment-Based Discovery of Potent and Selective DDR1/2 InhibitorsEnzymatic activity of Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors
All present enzymatic activity of Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors:
2.7.10.1; Protein crystallography data
The structure of Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors, PDB code: 5bvn
was solved by
C.Murray,
V.Berdini,
I.Buck,
M.Carr,
A.Cleasby,
J.Coyle,
J.Curry,
J.Day,
K.Hearn,
A.Iqbal,
L.Lee,
V.Martins,
P.Mortenson,
J.Munck,
L.Page,
S.Patel,
S.Roomans,
T.Kirsten,
G.Saxty,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Other elements in 5bvn:
The structure of Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors also contains other interesting chemical elements:
Fluorine Binding Sites:
The binding sites of Fluorine atom in the Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors
(pdb code 5bvn). This binding sites where shown within
5.0 Angstroms radius around Fluorine atom.
In total only one binding site of Fluorine was determined in the Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors, PDB code: 5bvn: Fluorine binding site 1 out of 1 in 5bvnGo back to Fluorine Binding Sites List in 5bvn
Fluorine binding site 1 out
of 1 in the Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors
Mono view Stereo pair view
Reference:
C.W.Murray,
V.Berdini,
I.M.Buck,
M.E.Carr,
A.Cleasby,
J.E.Coyle,
J.E.Curry,
J.E.Day,
P.J.Day,
K.Hearn,
A.Iqbal,
L.Y.Lee,
V.Martins,
P.N.Mortenson,
J.M.Munck,
L.W.Page,
S.Patel,
S.Roomans,
K.Smith,
E.Tamanini,
G.Saxty.
Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors. Acs Med.Chem.Lett. V. 6 798 2015.
Page generated: Thu Aug 1 08:22:45 2024
ISSN: ISSN 1948-5875 PubMed: 26191369 DOI: 10.1021/ACSMEDCHEMLETT.5B00143 |
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